Glixx Laboratories Inc
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Glixx Laboratorie
CAS: 3033576-12-1
Chemical Name: N-(1-(1,1-Di(pyridin-2-yl)ethyl)-6-(1-methyl-6-oxo-5-(piperidin-4-ylamino)-1,6-dihydropyridin-3-yl)-1H-indol-4-yl)ethanesulfonamide
For Lab R&D Uses Only
Purity: >98% (HPLC)
Novel potent BD1-selective BET inhibitor with a Kd of 8.9 nM and 185-fold BD1/BD2 selectivity
Reference:
https://pubs.acs.org/doi/10.1021/acs.jmedchem.3c01837
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