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H3R/S1R antagonist KSK68

 

CAS: 2566715-91-9

 

Chemical Name: Cyclopropyl(4-(3-(4-(pyridin-4-yl)piperidin-1-yl)propoxy)phenyl)methanone

 

 
GLXC-29196For Lab R&D Uses Only
        Cat No: GLXC-29196

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Novel dual sigma and histamine H3 receptor antagonist, (H3R: Ki = 7.7 nM, sigma-1: Ki =3.6 nM and sigma-2: Ki = 22.4 nM)

 

Reference:

https://pubs.acs.org/doi/10.1021/acs.jmedchem.3c00430

 

Analytical data click for PDF file

 

 

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