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INCB159020

 

CAS: 2923669-20-7

 

Chemical Name: 3-(1-((1R,4R,5S)-2-Azabicyclo[2.1.1]hexan-5-yl)-7-(3-chloro-2-methylphenyl)-6-fluoro-4-(5-methylpyrazin-2-yl)-2-((R)-1-(3-oxomorpholino)ethyl)-1H-pyrrolo[3,2-c]quinolin-8-yl)propanenitrile

 

 
GLXC-29277For Lab R&D Uses Only
        Cat No: GLXC-29277

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Novel potent KRAS G12D inhibitor (SPR kd=2.2 nM) for treating KRAS-driven cancers

 

Reference:

https://pubs.acs.org/doi/10.1021/acs.jmedchem.4c02662

 

Analytical data click for PDF file

 

 

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