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CAS: 2736508-65-7
Chemical Name: 3-tert-Butyl-N-[(1R)-1-[4-[6-[5-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide
For Lab R&D Uses Only
Purity: >98% (HPLC)
Novel BTK degrader, significantly reducing BTK protein levels in both peripheral blood and tumor tissue
References:
https://bpspubs.onlinelibrary.wiley.com/doi/10.1111/bph.17332
https://www.nature.com/articles/s41375-024-02317-4
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