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CAS: 3104736-80-0
Chemical Name: 4-(4-Chloro-2-((4-chloro-3-(trifluoromethyl)phenyl)sulfonamido)phenoxy)-N-(6-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)amino)hexyl)benzamide
For Lab R&D Uses Only
Purity: >98% (HPLC)
The first CCR2 molecular degrader, displaying sustained and concentration-dependent degradation of CCR2 over 24 h, efficiently inhibiting monocyte migration in a transwell assay
Reference:
https://pubs.acs.org/doi/10.1021/acs.jmedchem.5c02920
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