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CAS: 3065121-94-7
Chemical Name: 5-(3-Ethyl-4-((4-fluorobenzyl)amino)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-6-yl)benzo[c][1,2]oxaborol-1(3H)-ol
For Lab R&D Uses Only
Purity: >98% (HPLC)
Novel potent inhibitor of Cryptosporidium against the parasite in a cell-based infection model (EC50 = 0.19 μM) and non-cytotoxic, having a fast rate of parasite-killing and being orally efficacious in a Cryptosporidium mouse infection model (50 mg/kg BID)
Reference:
https://pubs.acs.org/doi/10.1021/acs.jmedchem.4c02805
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