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CAS: 2227484-71-9
Chemical Name: 2-((3-Amino-5H-pyrrolo[2,3-b]pyrazine-2-carboxamido)methyl)-5-(4-(bis((2S,3R,4R,5R)-2,3,4,5,6-pentahydroxyhexyl)amino)piperidine-1-carbonyl)-1,3-diethyl-1H-benzo[d]imidazol-3-ium trifluoroacetate TFA salt
For Lab R&D Uses Only
Purity: >98% (HPLC)
Novel inhibitor of RNA polymerase I, causing nucleolar stress and showing potent anticancer activity across many tumor types
References:
https://www.sciencedirect.com/science/article/pii/S022352342400922X
https://www.cysticfibrosisjournal.com/article/S1569-1993(24)00081-X/fulltext
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