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CAS: 3060519-94-7
Chemical Name: (E)-N1-(2-(3-(6,7-Dichloro-2-(2-hydroxyacetyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indol-9-yl)-1H-pyrazol-1-yl)ethyl)-N11-(2-(5-(4-(4-(dimethylamino)but-2-enoyl)-2-oxopiperazin-1-yl)thiophen-2-yl)ethyl)undecanediamide
For Lab R&D Uses Only
Purity: >98% (HPLC)
First-in-class Deubiquitinase-targeting Chimera (DUBTAC) of cGAS, effectively stabilizing cGAS and activated the cGAS/STING/IRF3 signaling
Reference:
https://onlinelibrary.wiley.com/doi/10.1002/anie.202415168
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