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CAS: N/A
Chemical Name: 4-((7-Acryloyl-2,7-diazaspiro[4.4]nonan-2-yl)methyl)-N-(2-(2-((S)-4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)acetamido)ethyl)-benzamide
For Lab R&D Uses Only
Purity: >98% (HPLC)
Novel covalent 14-3-3 molecular glue to sequester BRD4 into the cytosol
Reference:
https://pubs.acs.org/doi/10.1021/jacs.3c12389
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