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CAS: 2857845-45-3
Chemical Name: (2S,5S)-4-(3,3-Difluoro-2,2-dimethylpropanoyl)-2,3,4,5-tetrahydro-2,5-methanopyrido[3,4-f][1,4]oxazepine-9-carbonitrile
For Lab R&D Uses Only
Purity: >98% (HPLC)
Novel CNS-penetrant allosteric RIPK1 inhibitor, a bridged derivative of Oditrasertib (GLXC-27896), blocking necroptotic cell death
Reference:
https://pubs.acs.org/doi/10.1021/acsmedchemlett.5c00063
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