Glixx Laboratories Inc

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MS182

 

CAS: 3034773-62-8

 

Chemical Name: N-(2-(4-(2-(5-(3,5-Dimethylisoxazol-4-yl)-1-(2-morpholinoethyl)-1H-benzo[d]imidazol-2-yl)ethyl)-2-fluorophenoxy)ethyl)-1-(9-ethyl-7-(4-methylthiophen-2-yl)-9H-carbazol-3-yl)-5,8,11-trioxa-2-azatetradecan-14-amide

 

 
GLXC-28800For Lab R&D Uses Only
        Cat No: GLXC-28800

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Novel p53Y220C AceTAC, effectively acetylating p53Y220C at lysine 382 in a time- and concentration-dependent manner via inducing the ternary complex formation between p300/CBP acetyltransferase and p53Y220C

 

Reference:

https://pubs.acs.org/doi/10.1021/acs.jmedchem.4c01497

 

Analytical data click for PDF file

 

 

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