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LRK-4189

 

CAS: 3063346-83-5

 

Chemical Name: (1S,4R)-4-(4-(4-(((S)-2,6-Dioxopiperidin-3-yl)amino)-2-fluorophenyl)piperazin-1-yl)-N-((1r,4R)-4-((5-fluoro-4-(3-(2-oxopyridin-1(2H)-yl)phenyl)pyrimidin-2-yl)amino)cyclohexyl)cyclohexane-1-carboxamide

 

 
GLXC-29605For Lab R&D Uses Only
        Cat No: GLXC-29605

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

First-in-class degrader of the lipid kinase PIP4K2C for the treatment of Microsatellite Stable (MSS) Colorectal Carcinoma

 

Reference:

https://acs.digitellinc.com/p/s/discovery-of-lrk-4189-a-first-in-class-degrader-of-the-lipid-kinase-pip4k2c-for-the-treatment-of-microsatellite-stable-mss-colorectal-carcinoma-640250

 

Analytical data click for PDF file

 

 

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