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CAS: N/A
Chemical Name: (S)-N-((2S,14S,Z)-14-Carbamoyl-3,12,17-trioxo-1-phenyl-7,10-dioxa-4,13,16-triazadotriacont-25-en-2-yl)-1-(3-(N-(4-chlorobenzyl)sulfamoyl)-4-methoxybenzoyl)pyrrolidine-2-carboxamide
For Lab R&D Uses Only
Purity: >98% (HPLC)
Novel modulator of mTORC2 pathway, selectively binding to mSin1PH, impairing mTORC2’s membrane interactions, resulting in reduced AKT1 phosphorylation
Reference:
https://pubs.acs.org/doi/10.1021/acschembio.4c00597
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