Glixx Laboratories Inc
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Glixx Laboratorie
CAS: 2980682-00-4
Chemical Name: 5-Cyclopropyl-2-N-(2,6-difluoro-4-methylsulfonylphenyl)-2-N-methyl-6-(1-methylimidazol-4-yl)-4-N-(5-methyl-1H-pyrazol-3-yl)pyrimidine-2,4-diamine
For Lab R&D Uses Only
Purity: >98% (HPLC)
First-in-class orally bioavailable, selective PLK4 inhibitor, demonstrating exquisite selectivity over related kinases, including AURKA/B and PLK1, disrupting centriole biogenesis in cancer cells, modulates pharmacodynamic readouts of PLK4 activity in xenograft tumor tissues, and being efficacious in multiple TRIM37-amplified xenograft models
Reference:
https://pubs.acs.org/doi/10.1021/acs.jmedchem.5c00529
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