Glixx Laboratories Inc
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Glixx Laboratorie
CAS: 2906968-72-5
Chemical Name: 4-(3-Fluoro-4-((2-oxo-3-(propan-2-ylidene)indoline)-5-sulfonamido)phenoxy)-N-methylpicolinamide
For Lab R&D Uses Only
Purity: >98% (HPLC)
Novel selective CDK8 inhibitor (IC50 of 129 nM), inhibiting TGF-β1-mediated Smad3/RNA pol II phosphorylation and Akt/GSK3β/β-catenin signaling, inhibiting prostate cancer metastasis in vitro and in vivo
References:
https://www.ijbs.com/v21p0685.htm
https://www.sciencedirect.com/science/article/pii/S0753332223004559
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