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CAS: 2906968-72-5

 

Chemical Name: 4-(3-Fluoro-4-((2-oxo-3-(propan-2-ylidene)indoline)-5-sulfonamido)phenoxy)-N-methylpicolinamide

 

 
GLXC-29504For Lab R&D Uses Only
        Cat No: GLXC-29504

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Novel selective CDK8 inhibitor (IC50 of 129 nM), inhibiting TGF-β1-mediated Smad3/RNA pol II phosphorylation and Akt/GSK3β/β-catenin signaling, inhibiting prostate cancer metastasis in vitro and in vivo

 

References:

https://www.ijbs.com/v21p0685.htm

https://www.sciencedirect.com/science/article/pii/S0753332223004559


Analytical data click for PDF file

 

 

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