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COS-2080

 

CAS: N/A

 

Chemical Name: 2-(3-(3-(Dimethylcarbamoyl)-6-fluoroimidazo[1,2-a]pyridin-2-yl)azetidin-1-yl)-N-((3-oxo-3H-1,2,4-dithiazol-5-yl)methyl)quinoline-4-carboxamide

 

 
GLXC-29117For Lab R&D Uses Only
        Cat No: GLXC-29117

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Novel carbonyl sulfide (COS)/hydrogen sulfide (H2S)-donor hybrid phosphodiesterase 10A (PDE10A) inhibitor, demonstrating significant antifibrotic effects by inhibiting cell proliferation and mitigating fibroblast-to-myofibroblast transition (FMT)

 

Reference:

https://pubs.acs.org/doi/10.1021/acsptsci.4c00671

 

Analytical data click for PDF file

 

 

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