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CAS: 2410796-89-1
Chemical Name: 2-(6-Azaspiro[2.5]octan-6-yl)-4-(2-hydroxyethylsulfonylamino)-N-[6-[(2R)-2-methylmorpholin-4-yl]pyridin-2-yl]benzamide
For Lab R&D Uses Only
Purity: >98% (HPLC)
Novel inhibitor of kinesin KIF18A, revealing a mitotic vulnerability enriched in chromosomally unstable cancers, showing cell potency relative to AM-7710 and exhibiting good specificity against a panel of diverse kinesin motor proteins, except for the KIF19A motor
Reference:
https://www.nature.com/articles/s43018-023-00699-5
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