Glixx Laboratories Inc

               Your exclusive source for bioactive molecules

Glixx Laboratorie

 

   sales@glixxlabs.com      Toll-Free: (855)Go-Glixx   Tel: 781-333-5348    Fax: 781-333-5368 
VU6036864

 

CAS: 2746406-36-8

 

Chemical Name: 5-[4-(7-Chloro-[1,2,4]triazolo[1,5-a]pyridin-6-yl)-2,2,6,6-tetradeuteriopiperidin-1-yl]sulfonyl-2-methyl-1,3-oxazole

 

 
For Lab R&D Uses Only
        Cat No: GLXC-28789

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Novel antagonist tool compound of the M5 muscarinic acetylcholine receptor, showing exquisite potency (human M5 IC50 = 20 nM), good subtype selectivity (>500 fold selectivity against human M1-4), desirable brain exposure (Kp = 0.68, Kp,uu = 0.65), and high oral bioavailability (%F > 100%)

 

Reference:

https://pubs.acs.org/doi/10.1021/acs.jmedchem.4c01193


Analytical data click for PDF file

 

 

Place an order!

Price & Availability





email us for best prices
 








inquiry contact:
sales@glixxlabs.com
service@glixxlabs.com