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CAS: N/A
Chemical Name: Phenyl (S)-2-methoxy-5-(4-((1-(tetrahydro-2H-pyran-4-carbonyl)pyrrolidin-3-yl)amino)pyrido[3,2-d]pyrimidin-6-yl)nicotinate
For Lab R&D Uses Only
Purity: >98% (HPLC)
Novel lysine-targeted covalent inhibitor of PI3Kδ, exhibiting potently antitumor efficacy without obvious toxicity in the SU-DHL-6 and Pfeiffer xenograft mouse models
Reference:
https://pubs.acs.org/doi/10.1021/acs.jmedchem.4c01284
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