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Glixx Laboratorie
CAS: N/A
Chemical Name: {D-Arg}KKRR{Orn}RRR{beta-Ala}WKHAVIFWGNDPYGLKK; D-Arg-Lys-Lys-Arg-Arg-Orn-Arg-Arg-Arg-beta-Ala-Trp-Lys-His-Ala-Val-Ile-Phe-Trp-Gly-Asn-Asp-Pro-Tyr-Gly-Leu-Lys-Lys
For Lab R&D Uses Only
Purity: >98% (HPLC)
Novel putative CHD4 inhibitor peptide, interacting with CHD4 at its PHD domain with a dissociation constant (KD) of 14 nM. inducing caspase-mediated CHD4 cleavage, triggering cell death, and inhibiting tumor growth in a xenograft mouse model
Reference:
https://www.cell.com/cell-chemical-biology/fulltext/S2451-9456(24)00438-0
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