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Glixx Laboratorie
CAS: 1883429-22-8
Chemical Name: 4-(4-Dimethylaminomethyl-2,5-dimethoxy-phenyl)-2-methyl-2H-[2,7]naphthyridin-1-one
Cat No: GLXC-07027
Purity: > 98% (HPLC)
Storage: Refrigerator (4 °C)
Novel BRD9/7 specific inhibitor, binding to BRD9 with a higher affinity (Kd=14 nM, ITC) than to BRD7 (Kd=239nM, ITC), being completely negative on BET family members (>100 µM by AlphaScreen) and demonstrating cellular activity by FRAP on BRD9 and BRD7 at 0.1 µM and 1 µM, respectively
References:
1) https://www.mdpi.com/1422-0067/18/7/1537
2) https://pubs.acs.org/doi/10.1021/acs.jmedchem.6b00550
3) https://pubs.acs.org/doi/10.1021/acs.jmedchem.5b01865
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