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CAS: N/A
Chemical Name: (2S,4R)-1-((2S)-2-(4-(4-((2-(6-((4-((4-Chloro-3-fluorophenyl)amino)-7-methoxyquinazolin-6-yl)oxy)hexanamido)-3-((6-(4-(2-fluoro-5-((4-oxo-3,4-dihydrophthalazin-1-yl)methyl)benzoyl)piperazin-1-yl)-6-oxohexyl)amino)-3-oxopropoxy)methyl)-1H-1,2,3-triazol-1-yl)butanamido)-3,3-dimethylbutanoyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide
Purity: >98% (HPLC)
Novel Dual PROTAC for Simultaneous Degradation of EGFR and PARP
Ref: https://pubs.acs.org/doi/10.1021/acs.jmedchem.1c00649
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