Glixx Laboratories Inc

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Glixx Laboratorie

 

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ZL3138

 

CAS: N/A

 

Chemical Name: (S)-2-((1-(3-(4-(tert-Butyl)cyclohexyl)-4-(pyrrolidin-3-yloxy)benzoyl)piperidin-4-yl)oxy)-4-(piperazin-1-yl)benzonitrile dihydrochloride

 

 
GLXC-24310For Lab R&D Uses Only
        Cat No: GLXC-24310

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Novel β-catenin/B-cell lymphoma 9 (BCL9) inhibitor, disrupting the β-catenin/BCL9 protein-protein interaction (PPI) with a Ki of 0.96 μM and without affecting the β-catenin/E-cadherin interaction in living cells, displaying good selectivity for β-catenin/BCL9 over β-catenin/E-cadherin PPIs

 

Ref: https://pubs.acs.org/doi/10.1021/acs.jmedchem.1c00596

 

Analytical data click for PDF file

 

 

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