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RK-582

 

CAS: 2171388-28-4

 

Chemical Name: 6-((2R,6S)-2,6-Dimethylmorpholino)-4-fluoro-1-methyl-1'-(8-methyl-4-oxo-3,4,5,6,7,8-hexahydropyrido[2,3-d]pyrimidin-2-yl)spiro[indoline-3,4'-piperidin]-2-one

 

 
GLXC-22503For Lab R&D Uses Only
        Cat No: GLXC-22503

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Novel highly selective, potent tankyrase (TNKS/TNKS2) inhibitor, exhibiting a markedly improved robust tumor growth inhibition in a COLO-320DM mouse xenograft model

 

Ref: https://pubs.acs.org/doi/10.1021/acs.jmedchem.0c00045

 

Analytical data click for PDF file

 

 

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