Glixx Laboratories Inc
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Glixx Laboratorie
CAS: 2140301-96-6
Chemical Name: Brepocitinib tosylate; [(1S)-2,2-Difluorocyclopropyl][3-[2-[(1-methyl-1H-pyrazol-4-yl)amino]-4-pyrimidinyl]-3,8-diazabicyclo[3.2.1]oct-8-yl]-methanone tosylate
Purity: >98% (HPLC)
Novel inhibitor of JAK1 and TYK2 kinases, preventing IL-23 (interleukin 23) signaling through TYK2 (Tyrosine-protein kinase 2)/JAK1 (Janus kinase 1) inhibition
References:
1) https://pubs.acs.org/doi/10.1021/acs.jmedchem.8b00917
2) https://www.ncbi.nlm.nih.gov/pubmed/29266308
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