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CAS: N/A
Chemical Name: 6-(4-(2-((7-(4-(5-(Acrylamidomethyl)-4,5-dihydroisoxazol-3-yl)-2-fluorophenoxy)heptyl)amino)-2-oxoethyl)piperazin-1-yl)-N-(4-(3-chloro-4-cyanophenoxy)cyclohexyl)pyridazine-3-carboxamide
Purity: >98% (HPLC)
Novel androgen receptor (AR) degrader through E2 recruitment
Reference:
https://pubs.acs.org/doi/10.1021/acschembio.3c00040
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