Glixx Laboratories Inc
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Glixx Laboratorie
CAS: 2245231-10-9
Chemical Name: (2S)-2-[4-(4-Chlorophenyl)-2,3,6-trimethyl-1-[(1-methylpyrazol-4-yl)methyl]pyrrolo[2,3-b]pyridin-5-yl]-2-[(2-methylpropan-2-yl)oxy]acetic acid
For Lab R&D Uses Only
Purity: >98% (HPLC)
First-in-class inhibitor of allosteric integrase (ALLINI), targeting LEDGF/p75 binding site, displaying picomolar IC50 in human PBMCs with a >24,000 therapeutic index against HIV-1
Reference:
https://journals.asm.org/doi/full/10.1128/mbio.03560-22
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