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CAS: N/A
Chemical Name: 1-((1S,3r)-3-(4-(2-chlorophenyl)-5-(pyrimidin-4-yl)-4H-1,2,4-triazol-3-yl)cyclobutyl)-2-oxo-2,3-dihydro-1H-benzo[d]imidazole-5-carbonitrile
Purity: >98% (HPLC)
Novel potent and selective tankyrase inhibitor (TNKS1: 29 nM and TNKS2: 6.3 nM)
Ref: https://jeccr.biomedcentral.com/articles/10.1186/s13046-021-01950-6
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