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CAS: N/A
Chemical Name: 1-[(3R)-3-[2-[4-Hydroxy-1-[(2R,3S)-2-propyl-1-[3-(trifluoromethyl)pyridine-2-carbonyl]-3-[5-(trifluoromethyl)thiophen-3-yl]oxypiperidine-3-carbonyl]piperidin-4-yl]phenoxy]butyl]cyclobutane-1-carboxylic acid
Purity: >98% (HPLC)
Novel MDM2 Inhibitor, stabilizing the tumor suppressor TP53 and inducing growth arrest or apoptosis downstream of TP53 induction
References:
1) https://www.sciencedirect.com/science/article/abs/pii/S0223523422002367
2) https://www.sciencedirect.com/science/article/abs/pii/S022352341830816X
3) https://ascopubs.org/doi/10.1200/JCO.2016.70.7117
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