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Glixx Laboratorie
CAS: N/A
Chemical Name: N-(3-((6-Fluoro-2-((4-(4-methylpiperazin-1-yl)phenyl)amino)quinazolin-4-yl)amino)phenyl)acrylamide
Purity: >98% (HPLC)
Novel selective EGFR L858R/T790M inhibitor, exhibiting strong inhibitory activity against EGFR L858R/T790M (IC50 = 3.5 nM) and greater than 368-fold selectivity over EGFR WT (IC50 = 1290 nM), a 6.7-fold improvement over osimertinib, effectively inhibiting downstream signaling pathways and inducing apoptosis in mutant cells
Reference:
https://pubs.acs.org/doi/10.1021/acs.jmedchem.3c00027
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