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CAS: 1581714-49-9
Chemical Name: PRN473; (E)-2-[(3R)-3-[4-Amino-3-(2-fluoro-4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidine-1-carbonyl]-4,4-dimethylpent-2-enenitrile
Purity: >98% (HPLC)
Novel covalent reversible BTK inhibitor, exhibiting potent and durable inhibition of BTK, in vivo efficacy in rodent arthritis models, and clinical efficacy in canine pemphigus foliaceus
References:
https://pubmed.ncbi.nlm.nih.gov/?term=PRN473&sort=date
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