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CAS: 2723568-72-5
Chemical Name: FAP-targeted PI3Ki; N-(4-(((4-(((S)-1-((S)-2-Cyano-4,4-difluoropyrrolidin-1-yl)-1-oxopropan-2-yl)carbamoyl)pyridin-2-yl)methyl)amino)-4-oxobutanoyl)-S-((2-((((5-(6-(5-((2,4-difluorophenyl)sulfonamido)-6-methoxypyridin-3-yl)quinolin-4-yl)pyridin-2-yl)methoxy)carbonyl)oxy)ethyl)thio)cysteine
Purity: >98% (HPLC)
Novel FAP-targeted PI3K inhibitor, suppressing phosphorylation of Akt in IPF fibroblasts
Ref: https://stm.sciencemag.org/content/12/567/eaay3724
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