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CAS: N/A
Chemical Name: (S)-2-(3-(5-(2-(5-Isopropyl-2-methylphenoxy)pyrimidin-4-yl)-4-(4-(trifluoromethyl)phenyl)-1H-imidazol-1-yl)pyrrolidin-1-yl)-N,N-dimethylethan-1-amine
Purity: >98% (HPLC)
Novel potent BRD4 D1 inhibitor with over 500-fold selectivity against BRD2 D1 and BRD4 D2 via ITC
Ref: https://pubs.acs.org/doi/10.1021/acs.jmedchem.1c01779
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