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Glixx Laboratorie
CAS: N/A
Chemical Name: (E)-15,22-Dioxa-4,11-diaza-5(2,5)-thiadiazola-10(3,6)-pyridazina-1,14(1,3)-dibenzenacyclodocosaphan-18-ene-3,12-dione
For Lab R&D Uses Only
Purity: >98% (HPLC)
Novel inhibitor of glutaminase 1 (GLS1) with high binding affinity (SPR, Kd = 24 nM; ITC, Kd = 37 nM), exhibiting a similar in vivo antitumor activity as CB839 (GLXC-06047)
Ref: https://pubs.acs.org/doi/10.1021/acs.jmedchem.0c02044
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