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CAS: 2412055-93-5
Chemical Name: 2-(2,6-Dioxopiperidin-3-yl)-4-((2-(3-(4-(6-(6-((R)-2-(3-fluorophenyl)pyrrolidin-1-yl)imidazo[1,2-b]pyridazin-3-yl)pyridin-2-yl)piperazin-1-yl)-3-oxopropoxy)ethyl)amino)isoindoline-1,3-dione
Purity: >98% (HPLC)
First-in-class tropomyosin receptor kinase (TRK) degrader, targeting the intracellular kinase domain of TRK
Ref: https://pubs.acs.org/doi/10.1021/acs.jmedchem.0c01342
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