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CAS: N/A
Chemical Name: N-(4-(2-(((3R)-1-((1-(2-(2,6-Dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindolin-5-yl)piperidin-4-yl)methyl)pyrrolidin-3-yl)oxy)pyrimidin-5-yl)phenyl)-N-((1r,4R)-4-((4-(5-(methylsulfonyl)pyridin-3-yl)-5-(trifluoromethyl)pyrimidin-2-yl)amino)cyclohexyl)acetamide
For Lab R&D Uses Only
Purity: >98% (HPLC)
Novel Potent, Orally Bioavailable, and Highly Selective CDK12/13 Dual Degrader for the Treatment of Triple-Negative Breast Cancer
Reference:
https://pubs.acs.org/doi/10.1021/acs.jmedchem.5c02232
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