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CAS: 1872436-42-4
Chemical Name: 2-Methoxybenzyl (S)-6-chloro-2'-methyl-6'-oxo-1'-(((R)-tetrahydrofuran-2-yl)methyl)-1',4',5',6'-tetrahydro-[3,4'-bipyridine]-3'-carboxylate
Purity: >98% (HPLC)
Novel Potent Agonist of the Bile Acid Receptor TGR5 (EC50: hTGR5 2 nM; mTGR5 3 nM)
Reference:
https://pubs.acs.org/doi/10.1021/acs.jmedchem.2c01881
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