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CAS: N/A
Chemical Name: CAF-382; N-(5-(((5-Isopropyloxazol-2-yl)methyl)thio)thiazol-2-yl)piperidine-4-carboxamide
For Lab R&D Uses Only
Purity: >98% (HPLC)
Novel potent and cell-active inhibitor of cyclin-dependent kinase-like 5 (CDKL5), also targeting several cyclin-dependent kinases (CDK9, CDK16, CDK17, and CDK18)
References:
https://pubs.acs.org/doi/10.1021/acsmedchemlett.4c00219
https://elifesciences.org/articles/88206
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