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Glixx Laboratorie
CAS: 2407452-77-9
Chemical Name: N-[5-[2-Fluoro-5-[[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethyl]carbamoyl]phenyl]-2-[(3S,5R)-3,4,5-trimethylpiperazin-1-yl]phenyl]-6-oxo-4-(trifluoromethyl)-1H-pyridine-3-carboxamide
Purity: >98% (HPLC)
Novel selective WDR5 degrader, inhibiting acute myeloid leukemia in patient-derived mouse models
Reference:
https://www.science.org/doi/10.1126/scitranslmed.abj1578
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