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G9a degrader G9D-4

 

CAS: N/A

 

Chemical Name: 4-(4-((2-Cyclohexyl-6-methoxy-7-(3-(pyrrolidin-1-yl)propoxy)quinazolin-4-yl)amino)piperidin-1-yl)-N-(8-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)amino)octyl)butanamide

 

 
GLXC-28827For Lab R&D Uses Only
        Cat No: GLXC-28827

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Novel selective G9a degrader, exhibiting effective antiproliferative activities in a panel of pancreatic cancer cell lines and being able to sensitize KRASG12D mutant pancreatic cancer cells to KRASG12D inhibitor MRTX1133

 

Reference:

https://pubs.acs.org/doi/10.1021/acs.jmedchem.4c01192

 

Analytical data click for PDF file

 

 

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