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CAS: N/A
Chemical Name: 4-(4-((2-Cyclohexyl-6-methoxy-7-(3-(pyrrolidin-1-yl)propoxy)quinazolin-4-yl)amino)piperidin-1-yl)-N-(8-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)amino)octyl)butanamide
Purity: >98% (HPLC)
Novel selective G9a degrader, exhibiting effective antiproliferative activities in a panel of pancreatic cancer cell lines and being able to sensitize KRASG12D mutant pancreatic cancer cells to KRASG12D inhibitor MRTX1133
Reference:
https://pubs.acs.org/doi/10.1021/acs.jmedchem.4c01192
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