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Glixx Laboratorie
CAS: 2892720-11-3
Chemical Name: (4-Amino-4-methylpiperidin-1-yl)(5-((2,3-dichlorophenyl)thio)furan-2-yl)methanone
Purity: >98% (HPLC)
Novel SHP2 allosteric inhibitor, demonstrating potent binding affinity (KD = 0.29 μM), enzymatic activity (IC50 = 1.2 μM) and similar binding interactions to SHP099
Reference:
https://pubs.acs.org/doi/10.1021/acs.jmedchem.4c01217
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