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CAS: N/A
Chemical Name: 3-(6-((1H-Imidazol-1-yl)sulfonyl)-1-oxoisoindolin-2-yl)piperidine-2,6-dione
Purity: >98% (HPLC)
Novel covalent blocker of the CRBN binding site, possessing excellent metabolic stability in human plasma, liver microsomes, and hepatocytes
Reference:
https://pubs.acs.org/doi/10.1021/acsmedchemlett.3c00371
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