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CAS: N/A
Chemical Name: (E)-3-Cyclopropyl-N-[(S)-(4,4-difluorocyclohexyl)-[7-[(1S)-2-methoxy-1-[(4S)-2-oxo-4-(trifluoromethyl)imidazolidin-1-yl]ethyl]imidazo[1,2-b]pyridazin-2-yl]methyl]-2-fluoroprop-2-enamide
For Lab R&D Uses Only
Purity: >98% (HPLC)
Novel potent IL-17 Inhibitor ( IL-17A IC50: 13 nM), effectively reducing knee swelling in a rat arthritis model
Reference:
https://pubs.acs.org/doi/10.1021/acs.jmedchem.4c01520
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