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CAS: N/A
Chemical Name: 2-(1-(2-Chloro-6-fluorobenzyl)-1H-pyrrolo[2,3-b]pyridin-3-yl)-5-cyclopropylpyrimidin-4-amine
Purity: >98% (HPLC)
Novel potent inhibitor of hDHODH (IC50 = 173.4 nM), exerting better therapeutic effects on ulcerative colitis than hDHODH inhibitor vidofludimus (GLXC-90163) and Janus kinase (JAK) inhibitor tofacitinib (GLXC-90059)
Reference:
https://pubs.acs.org/doi/10.1021/acs.jmedchem.3c01365
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