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hDHODH inhibitor w2

 

CAS: N/A

 

Chemical Name: 2-(1-(2-Chloro-6-fluorobenzyl)-1H-pyrrolo[2,3-b]pyridin-3-yl)-5-cyclopropylpyrimidin-4-amine

 

 
GLXC-27847For Lab R&D Uses Only
        Cat No: GLXC-27847

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Novel potent inhibitor of hDHODH (IC50 = 173.4 nM), exerting better therapeutic effects on ulcerative colitis than hDHODH inhibitor vidofludimus (GLXC-90163) and Janus kinase (JAK) inhibitor tofacitinib (GLXC-90059)

 

Reference:

https://pubs.acs.org/doi/10.1021/acs.jmedchem.3c01365

 

Analytical data click for PDF file

 

 

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