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COP1-ATGL modulator 86

 

CAS: 2946701-09-1

 

Chemical Name: 1-(3-Acetylphenyl)-3-(3-(2-methoxyethyl)-2,4-dioxo-1-(2-(piperidin-1-yl)ethyl)-1,2,3,4-tetrahydroquinazolin-6-yl)urea

 

 
GLXC-28044For Lab R&D Uses Only
        Cat No: GLXC-28044

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Novel COP1-ATGL modulator, increasing ATGL protein expression, reducing ATGL ubiquitination and COP1 autoubiquitination, and diminishing lipid accumulation in hepatocytes in the nanomolar range, abrogating triglyceride accumulation and resolved fibrosis in preclinical Nonalcoholic Fatty Liver Disease (NAFLD) model

 

Reference:

https://pubs.acs.org/doi/10.1021/acs.jmedchem.3c01431

 

Analytical data click for PDF file

 

 

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