Glixx Laboratories Inc
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Glixx Laboratorie
CAS: 2946701-09-1
Chemical Name: 1-(3-Acetylphenyl)-3-(3-(2-methoxyethyl)-2,4-dioxo-1-(2-(piperidin-1-yl)ethyl)-1,2,3,4-tetrahydroquinazolin-6-yl)urea
Purity: >98% (HPLC)
Novel COP1-ATGL modulator, increasing ATGL protein expression, reducing ATGL ubiquitination and COP1 autoubiquitination, and diminishing lipid accumulation in hepatocytes in the nanomolar range, abrogating triglyceride accumulation and resolved fibrosis in preclinical Nonalcoholic Fatty Liver Disease (NAFLD) model
Reference:
https://pubs.acs.org/doi/10.1021/acs.jmedchem.3c01431
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