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CAS: 2417408-46-7
Chemical Name: N-(4-((2-(4-(6-((6-Acetyl-8-cyclopentyl-5-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl)amino)pyridin-3-yl)piperazin-1-yl)-2-oxoethyl)amino)butyl)-2-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)oxy)acetamide
Purity: >98% (HPLC)
Novel selective CDK6 degrader, effectively inhibiting RB phosphorylation and FOXM1 expression
References:
https://www.mdpi.com/2073-4425/12/9/1355
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