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Glixx Laboratorie
CAS: 2750709-91-0
Chemical Name: KIN-3248; 1-((3S,5R)-1-Acryloyl-5-(methoxymethyl)pyrrolidin-3-yl)-3-((1-cyclopropyl-4,6-difluoro-1H-benzo[d]imidazol-5-yl)ethynyl)-5-(methylamino)-1H-pyrazole-4-carboxamide
Purity: >98% (HPLC)
Novel irreversible pan-FGFR tyrosine kinase inhibitor, overcoming FGFR resistance
References:
https://pubs.acs.org/doi/10.1021/acs.jmedchem.3c01819
https://ascopubs.org/doi/10.1200/JCO.2022.40.4_suppl.461
https://ascopubs.org/doi/10.1200/JCO.2023.41.4_suppl.TPS637
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9523489/
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