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CAS: 2944101-99-7
Chemical Name: 4-(4-Fluoro-3-(4-(4-(2-(6-oxo-3-(pyridin-3-yl)pyridazin-1(6H)-yl)ethoxy)quinolin-7-yl)piperazine-1-carbonyl)benzyl)phthalazin-1(2H)-one
Purity: >98% (HPLC)
Novel highly potent dual inhibitor, exhibiting excellent inhibitory activities against PARP1 (IC50 = 3.3 nM) and c-Met (IC50 = 32.2 nM), demonstrating good antiproliferative effects on HR-proficient cancer cell lines and those resistant to PARP1 inhibitors
Reference:
https://pubs.acs.org/doi/10.1021/acs.jmedchem.4c00077
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