Glixx Laboratories Inc

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C3TD879

 

CAS: 2850259-33-3

 

Chemical Name: (2R)-2-Amino-4,4-dimethyl-N-[3-methyl-4-(2-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl)phenyl]pentanamide

 

 
GLXC-28252For Lab R&D Uses Only
        Cat No: GLXC-28252

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

First-in-class citron kinase (CITK) chemical probe, potently inhibiting CITK catalytic activity (biochemical IC50 = 12 nM), binding directly to full-length human CITK in cells (NanoBRET Kd < 10 nM), and demonstrating favorable DMPK properties for in vivo evaluation

 

Reference:

https://pubs.acs.org/doi/10.1021/acs.jmedchem.3c01807

 

Analytical data click for PDF file

 

 

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