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CAS: N/A
Chemical Name: (Z)-N-((1r,4r)-4-((2-(Diethylamino)ethyl)carbamoyl)cyclohexyl)-34-methyl-4-oxa-2,9-diaza-1(4,2)-pyrimidina-3(1,3)-benzenacyclononaphan-6-ene-15-carboxamide
Purity: >98% (HPLC)
Novel potent macrocyclic MERTK/AXL dual inhibitor with good selectivity over TYRO3 and FLT3
Reference:
https://pubs.acs.org/doi/10.1021/acs.jmedchem.4c00148
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